Compounds > pd 153035

pd 153035 and N-[3-(trifluoromethyl)phenyl]-4-quinazolinamine

pd 153035 has been researched along with N-[3-(trifluoromethyl)phenyl]-4-quinazolinamine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bridges, AJ; Cody, DR; Denny, WA; Fry, DW; McMichael, A; Rewcastle, GW; Zhou, H1
Bridges, AJ; Cody, DR; Denny, WA; Fry, DW; Kraker, AJ; McMichael, A; Rewcastle, GW; Showalter, HD; Zhou, H1
Gallus, J; Juvale, K; Wiese, M1

Other Studies

3 other study(ies) available for pd 153035 and N-[3-(trifluoromethyl)phenyl]-4-quinazolinamine

ArticleYear
Tyrosine kinase inhibitors. 5. Synthesis and structure-activity relationships for 4-[(phenylmethyl)amino]- and 4-(phenylamino)quinazolines as potent adenosine 5'-triphosphate binding site inhibitors of the tyrosine kinase domain of the epidermal growth fa
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Adenosine Triphosphate; Amino Acid Sequence; ErbB Receptors; Humans; Molecular Sequence Data; Protein-Tyrosine Kinases; Quinazolines; Structure-Activity Relationship; Tumor Cells, Cultured; Type C Phospholipases

1995
Tyrosine kinase inhibitors. 8. An unusually steep structure-activity relationship for analogues of 4-(3-bromoanilino)-6,7-dimethoxyquinazoline (PD 153035), a potent inhibitor of the epidermal growth factor receptor.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Aniline Compounds; Binding Sites; Blotting, Western; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Humans; Kinetics; Molecular Conformation; Molecular Structure; Phosphorylation; Protein Binding; Quinazolines; Structure-Activity Relationship; Tumor Cells, Cultured

1996
Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2).
    Bioorganic & medicinal chemistry, 2013, Dec-15, Volume: 21, Issue:24

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Humans; Molecular Structure; Neoplasm Proteins; Quinazolines; Structure-Activity Relationship

2013